No abstract available
MeSH terms
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Amino Acid Sequence
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Animals
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Binding, Competitive
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COS Cells
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Guanidines
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Guinea Pigs
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Ileum / drug effects
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In Vitro Techniques
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Male
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Mice
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Models, Molecular
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Molecular Conformation
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Molecular Sequence Data
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Morphinans
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Muscle, Smooth / drug effects
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Mutation
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Naltrexone / analogs & derivatives*
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Naltrexone / chemical synthesis
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Naltrexone / metabolism
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Naltrexone / pharmacology
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Narcotic Antagonists / chemical synthesis*
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Narcotic Antagonists / metabolism
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Narcotic Antagonists / pharmacology
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Rats
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Receptors, Opioid, kappa / antagonists & inhibitors*
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Receptors, Opioid, kappa / metabolism
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Receptors, Opioid, mu / genetics*
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Receptors, Opioid, mu / metabolism*
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Vas Deferens / drug effects
Substances
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17-cyclopropylmethyl-6,7-didehydro-4,5-epoxy-5'-guanidinyl-3,14-dihydroxyindolo(2',3'-6,7)morphinan
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CNGN-TI compound
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Guanidines
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Morphinans
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Narcotic Antagonists
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Receptors, Opioid, kappa
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Receptors, Opioid, mu
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norbinaltorphimine
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Naltrexone